Publication Type

Journal Article

Journal Name

Phytochemistry

Publication Date

1-1-2003

Abstract

Five novel limonoids, 1-5, were isolated from the root bark of Turraea wakefieldii and were characterized as tecleaninoid derivatives. This is the first report of the natural occurrence of tecleanin-type limonoids with a five-membered-ring A-seco structure for which we propose the name neotecleanins. The relative stereochemical structures of compounds 1-5 were established on the basis of NMR spectroscopy. The absolute stereochemical structure of 5 was confirmed by X-ray diffraction methods. In mosquito larvicidal assays, compounds 1, 2 and 4 showed dose-dependent larvicidal activity against larvae of Anopheles gambiae s.s. © 2003 Elsevier Ltd. All rights reserved.

Keywords

Anopheles gambiae s.s, Larvicidal activity, Limonoids, Meliaceae, Neotecleanins, Tecleaninoids, Turraea wakefieldii

PubMed ID

14559274

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